DICYCLOMINE

Drugs in Pregnancy and Lactation.

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Name: DICYCLOMINE
Class: Parasympatholytic
Risk Factor:    BM

Fetal Risk Summary

This anticholinergic/antispasmodic agent was a component of a proprietary mixture (Bendectin, others) used for the treatment and prevention of pregnancy-induced nausea and vomiting from 1956 until 1976, when the product was reformulated. Dicyclomine was removed at that time because it was discovered that it did not contribute to the effectiveness of the mixture as an antiemetic (see also Doxylamine).

Animal studies conducted with dicyclomine alone, and in combination with doxylamine and pyridoxine (i.e., Bendectin), have found no evidence of impaired fertility or adverse fetal effects (1,2).

In the Collaborative Perinatal Project, 1,024 mother-child pairs of the 50,282 studied were exposed to dicyclomine during the 1st trimester (3, pp. 346–56). It was the most common parasympatholytic agent consumed by the women studied. A statistically significant association (standardized relative risk (SRR) 1.46) was discovered for minor malformations with 21 malformed children (3, p. 353). Other defects with an SRR greater than 1.5, and the number of affected newborns, were polydactyly in blacks (SRR 1.89; N=6; 277 black mothers), macrocephaly (SRR 8.8; N=3), diaphragmatic hernia (SRR 12.0; N=3), and clubfoot (SRR 1.8; N=7) (3, pp. 353, 477). For use anytime during pregnancy, 1,593 women consumed dicyclomine and an increased SRR was measured for macrocephaly (6.2; N=3) and pectus excavatum (1.8; N=9) (3, p. 492). The authors of this study, however, strongly cautioned that a causal relationship could not be inferred from any of these data, especially when the drug was used after the 1st trimester, and that independent confirmation was required with other studies.

A retrospective study published in 1971, involving more than 1,200 mothers, examined the relationship between drugs and congenital malformations (4). This investigation found that significantly fewer mothers of infants with major anomalies, as compared to normal controls, took antiemetics during the first 56 days of pregnancy. Dicyclomine was the fourth most frequently ingested antiemetic.

In a surveillance study of Michigan Medicaid recipients involving 229,101 completed pregnancies conducted between 1985 and 1992, 642 newborns had been exposed to dicyclomine during the 1st trimester (F. Rosa, personal communication, FDA, 1993). A total of 31 (4.8%) major birth defects were observed (27 expected). Specific data were available for six defect categories, including (observed/expected) 5/6 cardiovascular defects, 1/1 oral clefts, 0/0.5 spina bifida, 0/1 limb reduction defects, 0/2 hypospadias, and 3/1 hypospadias. Only with the latter defect is there a suggestion of a possible association, but other factors, including the mother's disease, concurrent drug use, and chance may be involved.

In summary, the use of dicyclomine during human pregnancy does not appear to represent a risk to the fetus or newborn. A 1990 review on the teratogenic risk of commonly used drugs categorized the risk from dicyclomine as “none” (5).

Breast Feeding Summary

No published reports on the excretion of dicyclomine into breast milk have been located. The manufacturer has received a case report of apnea in a breast-fed 12-day-old infant whose mother was receiving dicyclomine (personal communication, N.G. Dahl, Marion Merrell Dow, Inc., 1992). Following the adverse event, the mother was administered a single, 20-mg dose of the drug, and breast feeding was suspended for 24 hours. Plasma and milk concentrations of dicyclomine 2 hours after the dose were 59 ng/mL and 131 ng/mL (milk:plasma ratio 2.2), respectively. Although a causal relationship between dicyclomine and apnea was not established, similar adverse reactions have occurred when the drug was administered directly to infants (1). Consequently, dicyclomine should not be given to nursing women.

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World’s leading meds delivered to your door – and you don’t even need a prescription! Only certified, first class drugs on offer! Buy more and spend less with our great discount system.

References

  1. Product information. Bentyl. Marion Merrell Dow, Inc. 1992.
  2. Gibson JP, Staples RE, Larson EJ, Kuhn WL, Holtkamp DE, Newberne JW. Teratology and reproduction studies with an antinauseant. Toxicol Appl Pharmacol 1968;13:439–47.
  3. Heinonen OP, Slone D, Shapiro S. Birth Defects and Drugs in Pregnancy. Littleton, MA:Publishing Sciences Group, 1977.
  4. Nelson MM, Forfar JO. Associations between drugs administered during pregnancy and congenital abnormalities of the fetus. Br Med J 1971;1:523–7.
  5. Friedman JM, Little BB, Brent RL, Cordero JF, Hanson JW, Shepard TH. Potential human teratogenicity of frequently prescribed drugs. Obstet Gynecol 1990;75:594–9.

Index

Q&A about Dicyclomine

Tran N
Has anyone ever use dicyclomine for fun?
I was wondering if anyone ever used dicyclomine for fun, like how they use xanax pills, etc?
Darenkea...
You should NEVER use any kind of chemicals, pills or medications of any kind for recreation!

Do you not have a brain in your head???
glyw60
How does dicyclomine work as direct muscle relaxant? Blocking calcium? (Apart from anticholinergic effect)?
JD
Dicyclomine relieves spasms of the gastrointestinal tract (stomach and intestines) by blocking the actions of spasm-causing chemicals in the body.They prevent contraction of the muscles by blocking the acetylcholine receptors on the muscle cells. It blocks the receptor sites in the cells that use calcium to cause the spasm. by blocking the receptor no activity can occur
The Joker
How long should someone take Dicyclomine?
And is it used for Diverticulosis?
Jason Homan
Hi the Joker, many patients with diverticulosis have minimal or no symptoms, and do not require any specific treatment. A high fiber diet and fiber supplements are advisable to prevent constipation and the formation of more diverticula. The diverticulitis diet should be well balanced, but include high fibre foods such as fresh fruits, vegetables and whole grains. You should have plenty of water in your diverticulitis diet. Throw in half an hour exercise a day, and your bowel and digestive system should keep in good shape.

Patients with mild symptoms of bloating or abdominal pain may benefit from anti- spasmodic drugs such as chlordiazepoxide (Librax), dicyclomine (Bentyl), Donnatal, and hyoscyamine (Levsin). Some doctors also recommend avoidance of nuts, corn, seeds. To prevent complications of diverticulosis most likely, your doctor be recommend also to use oral antibiotics when symptoms are mild.

If diverticulitis has been diagnosed by your doctor, and is confirmed as a mild case, then your doctor will probably recommend some dietary changes, if you have symptoms more serious your doctor will probably recommend use drugs or surgical intervention.

You should take your doctor's advice.

Jason Homan
UR NEW MAN
what would happen if i accidentally took 5 dicyclomine 1omg capsules?
John de Witt
You can expect a mild-to-moderate anticholinergic toxidrome. Plug that one into your search engine and smoke it!.

Lee, I'm an emergency physician, and I almost always know more about treating overdoses than the person manning the phones at Poison Control. The nurses always seem to call anyway, though.
Dude 103
does dicyclomine tablets or Psyllium Powder cause colon cancer ?
also is Psyllium a laxative?

Please explain
Sabrina H
Dicyclomine HCL is prescribed for Irritable Bowel Syndrome that acts on nerve receptors to block Acetylcholine and the associated stimulation of the GI tract. Pysllium is a plant based fiber that forms bulk that stimulates GI motility and acts as a laxative. Psyllium isn't absorbed and thus has no systemic effects. Neither has any indication of causing cancer. Both do work on the GI tract, but in opposite ways.
pknapp10...
After taking dicyclomine for about 10 months, I find I am experiencing stomach cramps. Is this a side effect?
Spike
Typical side effects of dycylomine include dry mouth, blurred vision, confusion, agitation, increased heart rate, heart palpitations, constipation, difficulty urinating, and occasionally seizures can occur. Other potential side effects include changes in taste perception, difficulty swallowing, headache, nervousness, drowsiness, weakness, dizziness, impotence, flushing, difficulty falling asleep, nausea, vomiting, rash, bloating and difficulty breathing.

Stomach pain isn't generally recognized as a problem with dicyclomine.
miranda
how many dicyclomine is too many?
ive been taking 8 a day..one every 3 hrs

whne ur only suppost to take 4..one ever 6 hrs is that baddd?

or is it ok?
Inlove
Dicyclomine makes me trip out, even when I take one pill 4 times a day which is what the bottle says to do. Even when i take it as prescribed (4 a day) I feel extremely high and loopy. So I couldn't imagine taking more than that. I guess if you need it more often than 4 times a day you could take it, just make sure its not having an effect on your motor skills and such because it is a muscle relaxer.
mila j
is it safe to take dicyclomine 20 mg while pregnant?
i would prefer for a doctor or someone in the medical field to answer my question
Luken
You might be able to find out at www.drugs.com

Your doctor or pharmacist should be able to tell you.
Dude 103
Is Dicyclomine safe? What are the risks for taking this medication?
texjeff1...
Dicyclomine is called an anticholenergic used for stomach and intestinal cramps and spasms. It is a very old product and its side effects are more bothersome then serious: dry mouth, dry eyes and nose and drowsiness for the most part.
USArocks...
Does the drug "Bentyl" (Dicyclomine) help with nausea?
0
"Gentle Bentyl" is generally prescribed for irritable bowl syndrome which results in pain in the abdomen and relief from an irritated colon and its side-effects, such as diarrhea.

It is not an anti-emetic, or a condition such as nausea. However, one of its side effects is the reduction of nausea resulting from Crohns disease. So it may help, possibly not.

Nausea can be helped by avoiding food for awhile, drinking non-acidic, or caffeinated beverages. Pepto-Bismol, is one of the old standard treatments for an upset stomach.

If it continues for several hours, you need to be checked out because dehydration is a serious problem caused by this constant loss of fluids from your body.